SCHEMBL2778377

SCHEMBL2778377

COC(=O)c1c[nH]c2c(Cl)cc(C3CC(=O)N(Cc4ccccc4)C3=O)cc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.47
ALDH1A1 P00352 6/20 0.43
LMNA P02545 2/20 0.43
GPBAR1 Q8TDU6 3/20 0.43
GAA P10253 3/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42
CYP2C19 P33261 1/20 0.42
STAT6 P42226 1/20 0.42
GSK3B P49841 1/20 0.41
POLB P06746 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
TSHR P16473 2/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
ALOX15 P16050 1/20 0.40
KMT2A Q03164 2/20 0.39
MITF O75030 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2777419 0.87 NR4A2 (0.49) NR4A2ALDH1A1LMNAGPBAR1GAA
SCHEMBL2778056 0.85 NR4A2 (0.47) NR4A2ALDH1A1LMNAGPBAR1GAA
SCHEMBL985642 0.74 ALDH1A1 (0.43) ALDH1A1GPBAR1GAACYP1A2CYP3A4
SCHEMBL982774 0.74 GPBAR1 (0.41) ALDH1A1LMNAGPBAR1GAACYP1A2
SCHEMBL3602720 0.70 ALDH1A1 (0.59) ALDH1A1GAACYP1A2CYP3A4CYP2C9
SCHEMBL980864 0.69 GPBAR1 (0.42) ALDH1A1LMNAGPBAR1GAACYP1A2
SCHEMBL981418 0.69 ALDH1A1 (0.42) ALDH1A1LMNAGPBAR1GAACYP1A2
SCHEMBL29158183 0.68 GPBAR1 (0.59) ALDH1A1GPBAR1GAACYP1A2CYP3A4
SCHEMBL29158182 0.68 GPBAR1 (0.59) ALDH1A1GPBAR1GAACYP1A2CYP3A4
SCHEMBL2781955 0.68 NR4A2 (0.52) NR4A2ALDH1A1GPBAR1TSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257545-A1 PYRROLIDINYL DERIVATIVES AND USES THEREOF F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009115427-A1 PYRROLIDINYL DERIVATIVES AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2009-09-24 WO disclosed