SCHEMBL27784100

SCHEMBL27784100

CC(C)(C)OC(=O)[C@H](CN)c1nc(C(=O)O)co1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
C3AR1 Q16581 2/20 0.36
FBP1 P09467 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
PTPN1 P18031 1/20 0.31
LMNA P02545 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27784102 1.00 C3AR1 (0.36) C3AR1FBP1HDAC1HDAC8HDAC6
SCHEMBL28787203 1.00 C3AR1 (0.36) C3AR1FBP1HDAC1HDAC8HDAC6
SCHEMBL27979112 0.87 C3AR1 (0.35) C3AR1FBP1HDAC1HDAC8HDAC6
SCHEMBL3586133 0.82 C3AR1 (0.36) C3AR1FBP1HDAC1HDAC8HDAC6
SCHEMBL15214453 0.75 C3AR1 (0.43) C3AR1HDAC1HDAC8HDAC6LMNA
SCHEMBL27805940 0.74 POLB (0.31) LMNAKMT2A
SCHEMBL27805945 0.74 ABCB1 (0.41) HDAC1HDAC8HDAC6LMNAKMT2A
SCHEMBL27805943 0.74 ABCB1 (0.41) HDAC1HDAC8HDAC6LMNAKMT2A
SCHEMBL27805944 0.74 POLB (0.31) LMNAKMT2A
SCHEMBL800492 0.72 KMT2A (0.49) C3AR1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101768130-B Derivatives containing aminomethyl-5-membered aromatic heterocycle-4-carboxylic acid, preparation method, drug combination and application thereof TIANJIN INST PHARM RESEARCH 2012-07-04 CN disclosed
CN-101768130-A Derivatives containing aminomethyl-5-membered aromatic heterocycle-4-carboxylic acid, preparation method, drug combination and application thereof TIANJIN INST PHARM RESEARCH 2010-07-07 CN disclosed