SCHEMBL27979112

SCHEMBL27979112

COC(=O)c1coc([C@@H](CN)C(=O)OC(C)(C)C)n1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
C3AR1 Q16581 2/20 0.35
DAGLA Q9Y4D2 1/20 0.34
FBP1 P09467 1/20 0.33
CACNA1G O43497 3/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
HDAC1 Q13547 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28787203 0.87 C3AR1 (0.36) C3AR1FBP1HDAC1HDAC8HDAC6
SCHEMBL27784100 0.87 C3AR1 (0.36) C3AR1FBP1HDAC1HDAC8HDAC6
SCHEMBL27784102 0.87 C3AR1 (0.36) C3AR1FBP1HDAC1HDAC8HDAC6
SCHEMBL3583659 0.83 C3AR1 (0.35) C3AR1DAGLAFBP1CACNA1GSLC6A2
SCHEMBL15214452 0.77 C3AR1 (0.40) C3AR1DAGLA
SCHEMBL1196600 0.75 CACNA1G (0.38) DAGLAFBP1CACNA1GSLC6A2SLC6A4
SCHEMBL800494 0.74 KMT2A (0.48) C3AR1
SCHEMBL3511397 0.74 KMT2A (0.48) C3AR1
SCHEMBL12980639 0.74 C3AR1 (0.46) C3AR1
SCHEMBL10045822 0.74 C3AR1 (0.46) C3AR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104024258-A Pyrrolopyrazine kinase inhibitors HOFFMANN LA ROCHE 2014-09-03 CN disclosed