SCHEMBL2779286

SCHEMBL2779286

NC(=O)C1(C(=O)NCc2ccc(Nc3ccc(OCC(F)F)cc3C(F)(F)F)cc2)CC1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.34
CNR2 P34972 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
MGLL Q99685 1/20 0.33
ABHD6 Q9BV23 1/20 0.33
MET P08581 1/20 0.33
BTK Q06187 1/20 0.33
S1PR1 P21453 1/20 0.33
S1PR3 Q99500 1/20 0.33
HTR2A P28223 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
ACACB O00763 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2805728 0.99 PTGES (0.34) PTGESCNR2CA1CA2CA7
SCHEMBL2778630 0.89 NPC1 (0.40) CNR2BTK
Hydrochloric Acid SCHEMBL2805730 0.88 AKT2 (0.38) PTGESCNR2CA1CA2CA7
SCHEMBL2809865 0.87 TP53 (0.39) CNR2CA1CA2CA7CA9
SCHEMBL2781755 0.79 POLB (0.40) CA1CA2CA7CA9TRPV1
SCHEMBL13128518 0.79 BDKRB1 (0.45) PTGESCNR2BTKHTR2AACACB
SCHEMBL185482 0.78 MAOB (0.40) MGLLABHD6S1PR1S1PR3ACACB
SCHEMBL2808315 0.77 NPC1 (0.41) BTKS1PR1S1PR3
SCHEMBL13160207 0.77 BTK (0.32) BTK
SCHEMBL2809872 0.76 TP53 (0.40) CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed
WO-2010097372-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed