SCHEMBL27801351

SCHEMBL27801351

Cc1ccc(C#Cc2ccc(OC(F)F)c(C)c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
GRM5 P41594 1/20 0.37
CA12 O43570 2/20 0.36
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
CA9 Q16790 2/20 0.36
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
MAPT P10636 3/20 0.36
LMNA P02545 2/20 0.36
MAPK1 P28482 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
POLB P06746 1/20 0.36
AR P10275 1/20 0.36
KCNH2 Q12809 1/20 0.35
BACE1 P56817 4/20 0.35
REN P00797 1/20 0.35
CTSD P07339 1/20 0.35
CYP3A4 P08684 1/20 0.35
BACE2 Q9Y5Z0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4312620 0.93 BACE1 (0.37) ALDH1A1MEN1KMT2AMAPTBACE1
SCHEMBL4312471 0.89 BACE1 (0.40) GRM5MAPTARBACE1REN
SCHEMBL4306001 0.89 GRM5 (0.37) ALDH1A1GRM5MEN1KMT2AMAPT
SCHEMBL13932862 0.88 ALDH1A1 (0.38) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL4319022 0.86 GRM5 (0.44) ALDH1A1GRM5CA12CA1CA2
SCHEMBL4309762 0.84 BACE1 (0.38) ALDH1A1GRM5MEN1KMT2AMAPT
SCHEMBL27801226 0.81 FFAR1 (0.42) GRM5MEN1KMT2AARBACE1
SCHEMBL23190460 0.81 BACE1 (0.34) ALDH1A1MEN1KMT2AMAPTBACE1
SCHEMBL4313333 0.81 BACE1 (0.38) BACE1RENCTSDCYP3A4BACE2
SCHEMBL23190454 0.80 BACE1 (0.35) ALDH1A1GRM5MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101641335-A Amino-5-[substituted-4-(difluoromethoxy)phenyl]-5- phenylimidazolone compounds as ss-secretase inhibitors WYETH CORP US 2010-02-03 CN disclosed