SCHEMBL2780282

SCHEMBL2780282

CN(CCCN1CCCc2cc(NC(=N)c3cccs3)ccc21)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 10/20 0.51
NOS1 P29475 10/20 0.51
TP53 P04637 7/20 0.47
LMNA P02545 6/20 0.47
KCNH2 Q12809 3/20 0.46
MAPT P10636 2/20 0.44
POLB P06746 1/20 0.44
NOS2 P35228 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2675198 0.90 NOS3 (0.62) NOS3NOS1TP53LMNAKCNH2
SCHEMBL2675388 0.90 NOS3 (0.47) NOS3NOS1TP53LMNAKCNH2
SCHEMBL2675520 0.88 NOS3 (0.56) NOS3NOS1TP53LMNAKCNH2
SCHEMBL2675017 0.86 NOS3 (0.61) NOS3NOS1TP53LMNAKCNH2
SCHEMBL2675512 0.86 NOS3 (0.49) NOS3NOS1TP53LMNAKCNH2
SCHEMBL2677052 0.85 NOS3 (0.62) NOS3NOS1TP53LMNAKCNH2
SCHEMBL499211 0.84 NOS3 (0.52) NOS3NOS1MAPTNOS2MEN1
SCHEMBL2674397 0.84 TP53 (0.48) NOS3NOS1TP53LMNAKCNH2
SCHEMBL2676597 0.84 NOS3 (0.63) NOS3NOS1TP53LMNAKCNH2
SCHEMBL4112042 0.84 NOS3 (0.61) NOS3NOS1TP53LMNAKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139886-A1 QUINOLONE AND TETRAHYDROQUINOLINE AND RELATED COMPOUNDS HAVING NOS INHIBITORY ACTIVITY Neuraxon Inc. (CA) 2010-01-06 EP disclosed
WO-2008116308-A1 QUINOLONE AND TETRAHYDROQUINOLINE AND RELATED COMPOUNDS HAVING NOS INHIBITORY ACTIVITY NEURAXON, INC. (CA) 2008-10-02 WO disclosed