SCHEMBL27804848

SCHEMBL27804848

COc1cccc(C(O)c2ccc(NC(=O)C3(c4ccc5c(c4)OCO5)CC3)nc2)c1

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CFTR P13569 18/20 0.52
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27804842 0.90 CFTR (0.51) CFTRNPC1RAB9AKMT2A
SCHEMBL27825686 0.89 CFTR (0.50) CFTRNPC1RAB9AKMT2A
SCHEMBL27977473 0.87 CFTR (0.48) CFTR
SCHEMBL27804841 0.87 CFTR (0.48) CFTR
SCHEMBL27825584 0.86 CFTR (0.48) CFTR
SCHEMBL27825466 0.86 TP53 (0.48) CFTR
SCHEMBL1074831 0.85 CFTR (0.51) CFTRNPC1RAB9A
SCHEMBL27825454 0.85 CFTR (0.46) CFTRNPC1RAB9A
SCHEMBL27804844 0.85 CFTR (0.46) CFTR
SCHEMBL12188916 0.84 CFTR (0.58) CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103951614-A Pyridyl derivatives as CFTR modulators VERTEX PHARMA 2014-07-30 CN disclosed
CN-101981011-A Pyridyl derivatives as CFTR modulators VERTEX PHARMA 2011-02-23 CN disclosed