SCHEMBL27808293

SCHEMBL27808293

CC(=O)OCN(Cc1cccc(-c2cncc(-c3cc(-c4cccc(C)n4)nc4[nH]ccc34)c2)c1)C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C8 P10632 1/20 0.37
CDK8 P49336 6/20 0.33
ACACB O00763 1/20 0.33
JAK1 P23458 1/20 0.33
CFD P00746 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.31
TGFBR2 P37173 1/20 0.31
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31
CETP P11597 1/20 0.30
HDAC1 Q13547 1/20 0.30
PIKFYVE Q9Y2I7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3796758 0.90 CYP3A4 (0.38) TGFBR1CYP3A4CYP2C8ACACBJAK1
SCHEMBL4167086 0.89 CYP3A4 (0.38) TGFBR1CYP3A4CYP2C8CDK8ACACB
SCHEMBL27828792 0.89 TGFBR1 (0.36) TGFBR1CYP3A4CYP2C8CDK8ACACB
SCHEMBL27808283 0.87 TGFBR1 (0.39) TGFBR1CYP3A4CYP2C8CDK8JAK1
SCHEMBL27808284 0.84 TGFBR1 (0.42) TGFBR1CYP3A4CYP2C8CDK8JAK1
SCHEMBL27808346 0.82 TGFBR1 (0.37) TGFBR1CYP3A4CYP2C8IRAK4TGFBR2
SCHEMBL4156980 0.82 ACACB (0.43) TGFBR1CYP3A4CYP2C8CDK8ACACB
SCHEMBL27808216 0.81 TGFBR1 (0.40) TGFBR1CYP3A4CYP2C8CDK8JAK1
SCHEMBL27808359 0.81 TGFBR1 (0.39) TGFBR1CYP3A4CYP2C8CDK8JAK1
SCHEMBL4159244 0.80 TGFBR1 (0.45) TGFBR1CYP3A4CYP2C8CDK8TGFBR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101970435-A Pyrrolopyrimidines and pyrrolopyridines NOVARTIS AG 2011-02-09 CN disclosed