SCHEMBL27808352

SCHEMBL27808352

CC(=O)OCN(C)Cc1cccc(-c2cncc(-c3nc(-c4cccc(C)n4)nc4[nH]ccc34)c2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 3/20 0.39
TGFBR2 P37173 2/20 0.39
CDK8 P49336 8/20 0.35
PDK1 Q15118 3/20 0.33
MAP4K4 O95819 2/20 0.33
CHEK2 O96017 2/20 0.33
CDK1 P06493 2/20 0.33
FES P07332 2/20 0.33
ROS1 P08922 2/20 0.33
FER P16591 2/20 0.33
FLT4 P35916 2/20 0.33
KDR P35968 2/20 0.33
IRAK1 P51617 2/20 0.33
ROCK1 Q13464 2/20 0.33
PKN2 Q16513 2/20 0.33
MARK2 Q7KZI7 2/20 0.33
MINK1 Q8N4C8 2/20 0.33
AURKB Q96GD4 2/20 0.33
SLK Q9H2G2 2/20 0.33
MKNK2 Q9HBH9 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4150696 0.88 TGFBR1 (0.38) TGFBR1TGFBR2CDK8PDK1MAP4K4
SCHEMBL4165700 0.88 TGFBR1 (0.39) TGFBR1TGFBR2CDK8PDK1MAP4K4
SCHEMBL27828792 0.88 TGFBR1 (0.36) TGFBR1TGFBR2CDK8PDK1MAP4K4
SCHEMBL27808283 0.88 TGFBR1 (0.39) TGFBR1TGFBR2CDK8MAP4K4CHEK2
SCHEMBL3722712 0.86 TGFBR1 (0.39) TGFBR1TGFBR2CDK8PDK1CYP3A4
SCHEMBL4158616 0.86 TGFBR1 (0.42) TGFBR1TGFBR2CDK8CLK2CYP3A4
SCHEMBL28787418 0.86 TGFBR1 (0.40) TGFBR1TGFBR2CDK8MAP4K4CHEK2
SCHEMBL3672347 0.83 CDK8 (0.47) TGFBR1TGFBR2CDK8CYP3A4CYP2C8
SCHEMBL4301753 0.82 TGFBR1 (0.38) TGFBR1TGFBR2CDK8PDK1MAP4K4
SCHEMBL27808346 0.81 TGFBR1 (0.37) TGFBR1TGFBR2PDK1IRAK4CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101970435-A Pyrrolopyrimidines and pyrrolopyridines NOVARTIS AG 2011-02-09 CN disclosed