SCHEMBL27808992

SCHEMBL27808992

CCOC(=O)CC(=O)OCc1cccc(Br)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLA P06280 1/20 0.58
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C19 P33261 1/20 0.55
HCAR2 Q8TDS4 1/20 0.54
HSP90AA1 P07900 1/20 0.50
MMP1 P03956 1/20 0.50
MMP2 P08253 1/20 0.50
MMP9 P14780 1/20 0.50
MMP12 P39900 1/20 0.50
MAOB P27338 5/20 0.49
IDO1 P14902 2/20 0.47
AGXT P21549 2/20 0.47
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.47
MAOA P21397 1/20 0.46
PARP15 Q460N3 2/20 0.46
PARP14 Q460N5 1/20 0.46
PARP10 Q53GL7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20954673 0.86 GLA (0.59) GLACYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL7035447 0.84 HCAR2 (0.49) GLACYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL4137771 0.84 EGFR (0.47) GLACYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL788672 0.83 EGFR (0.48) GLAHCAR2MAOBMAPTGAA
SCHEMBL27972481 0.82 ALDH1A1 (0.55) CYP3A4HCAR2HSP90AA1MMP1MMP2
SCHEMBL4151444 0.81 TAAR1 (0.45) GLACYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL27787074 0.81 MAPT (0.56) MAPTMGAMGAASIMGAM2
SCHEMBL1557559 0.80 ALDH1A1 (0.61) MGAMGAASIMGAM2KMT2A
SCHEMBL24241987 0.80 CYP1A2 (0.56) GLACYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL1511063 0.80 CYP4F2 (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101784520-B Novel malonic acid sulfonamide derivative and pharmaceutical use thereof MITSUBISHI TANABE PHARMA CORP 2014-07-02 CN disclosed
CN-102791674-A Compound having trimethylene structure, polymer compound containing unit that has trimethylene structure, and reactive compound having trimethylene structure HITACHI CHEMICAL CO LTD 2012-11-21 CN disclosed
CN-101784520-A Novel malonic acid sulfonamide derivative and pharmaceutical use thereof MITSUBISHI TANABE PHARMA CORP 2010-07-21 CN disclosed