Mk-212

Mk-212

SCHEMBL27809059

CC(C)(C)OC=O.Clc1cncc(N2CCNCC2)n1

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.68
HTR2A P28223 4/20 0.68
ALDH1A1 P00352 2/20 0.68
HTR1A P08908 2/20 0.68
KDM4E B2RXH2 1/20 0.68
MEN1 O00255 1/20 0.68
CYP1A2 P05177 1/20 0.68
CYP3A4 P08684 1/20 0.68
CYP2C9 P11712 1/20 0.68
HPGD P15428 1/20 0.68
CYP2C19 P33261 1/20 0.68
KMT2A Q03164 1/20 0.68
HSD17B10 Q99714 1/20 0.68
HTR3A P46098 3/20 0.46
HTR3E A5X5Y0 2/20 0.46
HTR3B O95264 2/20 0.46
HTR3D Q70Z44 2/20 0.46
HTR3C Q8WXA8 2/20 0.46
HTR2B P41595 3/20 0.42
CHRM4 P08173 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tert-Butyl Formate SCHEMBL27829478 0.85 HTR2C (0.46) HTR2CHTR2AALDH1A1HTR1AKDM4E
Mk-212 SCHEMBL255453 0.82 HTR2A (1.00) HTR2CHTR2AALDH1A1HTR1AKDM4E
Mk-212 SCHEMBL29389957 0.82 HTR2A (1.00) HTR2CHTR2AALDH1A1HTR1AKDM4E
Mk-212 SCHEMBL3060615 0.81 HTR2A (0.96) HTR2CHTR2AALDH1A1HTR1AKDM4E
Mk-212 SCHEMBL12503246 0.79 HTR2A (0.93) HTR2CHTR2AALDH1A1HTR1AKDM4E
Tert-Butyl Formate SCHEMBL27896719 0.79 CNR2 (0.44) HTR2CHTR2AALDH1A1HTR1AKDM4E
Tert-Butyl Formate SCHEMBL27835002 0.78 ALDH1A1 (0.41) HTR2CHTR2AALDH1A1HTR1AKDM4E
SCHEMBL6360772 0.77 ALDH1A1 (0.87) HTR2CHTR2AALDH1A1HTR1AKDM4E
Tert-Butyl Formate SCHEMBL27815217 0.76 KDM4E (0.46) HTR2CHTR2AALDH1A1HTR1AKDM4E
Tert-Butyl Formate SCHEMBL27885957 0.76 KMT2A (0.44) HTR2CHTR2AALDH1A1HTR1AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102046601-B Benzene or thiophene derivative and use thereof as VAP-1 inhibitor R TECH UENO LTD 2014-08-27 CN disclosed
CN-102046601-A Benzene or thiophene derivative and use thereof as VAP-1 inhibitor R TECH UENO LTD 2011-05-04 CN disclosed