SCHEMBL27809063

SCHEMBL27809063

CN(C)c1ccc(C#Cc2c[c]ccc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
SNCA P37840 6/20 0.39
MAPT P10636 5/20 0.39
APP P05067 6/20 0.39
ADK P55263 5/20 0.38
ACACB O00763 1/20 0.36
GRM5 P41594 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2555531 0.78 APP (0.57) ALDH1A1ALOX15TSHRHSD17B10SNCA
SCHEMBL2188836 0.78 APP (0.57) ALDH1A1ALOX15TSHRHSD17B10MAPT
SCHEMBL770159 0.78 ALDH1A1 (0.65) ALDH1A1ALOX15TSHRHSD17B10SNCA
SCHEMBL10300053 0.78 ALDH1A1 (0.65) ALDH1A1ALOX15TSHRHSD17B10SNCA
SCHEMBL5496752 0.77 TSHR (0.46) ALDH1A1TSHRMAPTAPP
SCHEMBL5495027 0.76 APP (0.47) ALDH1A1ALOX15HSD17B10MAPTAPP
SCHEMBL5492434 0.76 MAPT (0.59) ALDH1A1HSD17B10MAPTAPPADK
SCHEMBL2539548 0.76 APP (0.37) MAPTAPPGRM5
SCHEMBL2545694 0.76 APP (0.37) MAPTAPP
SCHEMBL4268626 0.76 APP (0.37) MAPTAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102046601-A Benzene or thiophene derivative and use thereof as VAP-1 inhibitor R TECH UENO LTD 2011-05-04 CN disclosed