SCHEMBL27809191

SCHEMBL27809191

CC(=O)Nc1ccc(C#Cc2ccc(CNC(=O)NN)cc2)cn1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACACB O00763 15/20 0.44
PTK2 Q05397 1/20 0.43
PTPN1 P18031 1/20 0.42
AOC3 Q16853 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27981821 0.99 ACACB (0.43) ACACBPTK2PTPN1AOC3KDM4E
SCHEMBL27809002 0.88 ACACB (0.43) ACACBPTPN1AOC3KDM4EMEN1
Hydrochloric Acid SCHEMBL27981776 0.87 ACACB (0.43) ACACBPTPN1AOC3KDM4EMEN1
SCHEMBL1432897 0.84 RAB9A (0.44) ACACBPTK2AOC3KDM4EMEN1
SCHEMBL27808983 0.84 AOC3 (0.50) PTK2PTPN1AOC3
SCHEMBL27808962 0.83 RAB9A (0.61) PTPN1KDM4EMEN1ALDH1A1HPGD
Hydrochloric Acid SCHEMBL1432991 0.83 RAB9A (0.43) ACACBPTK2AOC3KDM4EMEN1
SCHEMBL27829450 0.83 EGLN1 (0.41) ACACBPTPN1AOC3KDM4EMEN1
Hydrochloric Acid SCHEMBL27981813 0.82 AOC3 (0.49) PTK2PTPN1AOC3
Hydrochloric Acid SCHEMBL27829482 0.82 RAB9A (0.59) PTPN1AOC3KDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102046601-A Benzene or thiophene derivative and use thereof as VAP-1 inhibitor R TECH UENO LTD 2011-05-04 CN claimed
CN-102046601-B Benzene or thiophene derivative and use thereof as VAP-1 inhibitor R TECH UENO LTD 2014-08-27 CN disclosed
CN-102046601-A Benzene or thiophene derivative and use thereof as VAP-1 inhibitor R TECH UENO LTD 2011-05-04 CN disclosed