SCHEMBL27818652

SCHEMBL27818652

CCC[C@@H](N(NC(=O)c1cc(C)cc(C)c1)C(=O)c1ccc(OC)c(OC)c1)C(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 4/20 0.42
TAS1R1 Q7RTX1 4/20 0.42
PKM P14618 1/20 0.41
ABCB1 P08183 4/20 0.41
CYP3A4 P08684 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC2 Q92769 1/20 0.40
SLC6A4 P31645 1/20 0.40
CTNNB1 P35222 2/20 0.39
WNT3A P56704 2/20 0.39
ELANE P08246 1/20 0.39
ALDH1A1 P00352 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2779356 0.96 TAS1R3 (0.44) TAS1R3TAS1R1PKMABCB1CYP3A4
SCHEMBL2682439 0.96 TAS1R3 (0.44) TAS1R3TAS1R1PKMABCB1CYP3A4
SCHEMBL2681891 0.90 ABCB1 (0.43) ABCB1CYP3A4
SCHEMBL2682545 0.90 ABCB1 (0.43) ABCB1CYP3A4
SCHEMBL19946436 0.90 ABCB1 (0.43) ABCB1CYP3A4
SCHEMBL27818653 0.90 ABCB1 (0.43) ABCB1CYP3A4
SCHEMBL28789040 0.86 ABCB1 (0.46) TAS1R3TAS1R1ABCB1CYP3A4
SCHEMBL2682521 0.85 ABCB1 (0.47) TAS1R3TAS1R1ABCB1CYP3A4
SCHEMBL14763701 0.85 ABCB1 (0.47) TAS1R3TAS1R1ABCB1CYP3A4
SCHEMBL27797503 0.84 ABCB1 (0.52) TAS1R3TAS1R1ABCB1CYP3A4SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101848887-A Chiral diacylhydrazine ligands for modulating exogenous gene expression via ecdysone receptor complexes INTREXON CORP 2010-09-29 CN claimed
CN-101848887-A Chiral diacylhydrazine ligands for modulating exogenous gene expression via ecdysone receptor complexes INTREXON CORP 2010-09-29 CN disclosed