SCHEMBL27830100

SCHEMBL27830100

CC(Nc1ncnc2ccccc12)c1cccc(NC(=O)C2CC2(C)C)c1

nearest known ligand 0.73

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AURKA O14965 17/20 0.73
RPS6KB1 P23443 16/20 0.73
AURKB Q96GD4 5/20 0.57
GALR3 O60755 1/20 0.54
NR2F2 P24468 1/20 0.54
ABCG2 Q9UNQ0 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27830098 1.00 AURKA (0.73) AURKARPS6KB1AURKBGALR3NR2F2
SCHEMBL665746 0.84 AURKA (1.00) AURKARPS6KB1AURKB
SCHEMBL665928 0.84 AURKA (1.00) AURKARPS6KB1AURKB
SCHEMBL665747 0.84 AURKA (1.00) AURKARPS6KB1AURKB
SCHEMBL665726 0.77 AURKA (1.00) AURKARPS6KB1AURKB
SCHEMBL664658 0.77 AURKA (1.00) AURKARPS6KB1AURKB
SCHEMBL665725 0.77 AURKA (1.00) AURKARPS6KB1AURKB
SCHEMBL27830110 0.75 AURKA (0.74) AURKARPS6KB1AURKBGALR3NR2F2
SCHEMBL27830081 0.74 AURKA (0.75) AURKARPS6KB1AURKB
SCHEMBL27848833 0.74 AURKA (0.76) AURKARPS6KB1AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102317269-A Novel amino aza heterocyclic carboxamides MERCK PATENT GMBH 2012-01-11 CN disclosed