SCHEMBL27848833

SCHEMBL27848833

CC(Nc1ncnc2ccccc12)c1cccc(NC(=O)c2ccc(N3CCN(C)CC3)cc2)c1

nearest known ligand 0.76

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AURKA O14965 18/20 0.76
RPS6KB1 P23443 17/20 0.76
AURKB Q96GD4 9/20 0.56
PDPK1 O15530 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL665444 0.86 AURKA (1.00) AURKARPS6KB1AURKBPDPK1
SCHEMBL28011761 0.82 AURKA (0.76) AURKARPS6KB1AURKB
SCHEMBL27830081 0.80 AURKA (0.75) AURKARPS6KB1AURKBPDPK1
SCHEMBL27830110 0.79 AURKA (0.74) AURKARPS6KB1AURKB
SCHEMBL666498 0.78 RPS6KB1 (0.85) AURKARPS6KB1AURKBPDPK1
SCHEMBL27830109 0.78 RPS6KB1 (0.75) AURKARPS6KB1AURKBPDPK1
SCHEMBL27848547 0.77 AURKA (0.75) AURKARPS6KB1AURKB
SCHEMBL28011763 0.76 GALR3 (0.47) AURKARPS6KB1AURKB
SCHEMBL27830100 0.74 AURKA (0.73) AURKARPS6KB1AURKB
SCHEMBL27830098 0.74 AURKA (0.73) AURKARPS6KB1AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102317269-A Novel amino aza heterocyclic carboxamides MERCK PATENT GMBH 2012-01-11 CN disclosed