Pyrimidine

Pyrimidine

SCHEMBL27835166

O=S(=O)(c1ccccc1)n1cc(Br)c2c(Cl)ccnc21.c1cncnc1

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.40
ENPP3 O14638 1/20 0.36
ENPP1 P22413 1/20 0.36
HTR6 P50406 6/20 0.36
PKM P14618 2/20 0.36
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
MET P08581 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33
CYP3A4 P08684 2/20 0.32
ABL1 P00519 1/20 0.32
BCR P11274 1/20 0.32
CYP3A5 P20815 1/20 0.32
HTR2A P28223 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2105176 0.94 CYP2C19 (0.45) CYP2C19ENPP3ENPP1HTR6PKM
SCHEMBL16023210 0.81 CA1 (0.47) HTR6PKMKDM4EALDH1A1GAA
SCHEMBL25278649 0.81 CA1 (0.47) HTR6PKMKDM4EALDH1A1GAA
SCHEMBL16050462 0.79 CYP2C19 (0.45) CYP2C19ENPP3ENPP1HTR6PKM
SCHEMBL1050296 0.79 CYP2C19 (0.45) CYP2C19ENPP3ENPP1HTR6PKM
SCHEMBL2253631 0.79 SRC (0.40) CYP2C19HTR6PKMMETALDH1A1
SCHEMBL2104972 0.76 CYP2C19 (0.42) CYP2C19ENPP3ENPP1HTR6PKM
SCHEMBL27815784 0.76 CYP2C19 (0.42) CYP2C19ENPP3ENPP1HTR6PKM
SCHEMBL2237471 0.75 LMNA (0.51) CYP2C19ENPP3ENPP1HTR6PKM
SCHEMBL20508781 0.74 HTT (0.43) CYP2C19HTR6PKMSMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102143746-A CDK modulators EXELIXIS INC 2011-08-03 CN disclosed