SCHEMBL27836799

SCHEMBL27836799

CS(=O)(=O)CCCOc1ncc2ccccc2n1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 7/20 0.39
TLR8 Q9NR97 6/20 0.38
CYP11B2 P19099 1/20 0.36
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP1A2 P05177 1/20 0.33
HTR3A P46098 1/20 0.33
HRH4 Q9H3N8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22579036 0.78 TLR8 (0.54) TLR8RAB9AKMT2ACYP1A2
SCHEMBL28691857 0.78 KDM4E (0.37) MKNK1TLR8HCRTR1HCRTR2KMT2A
SCHEMBL7044155 0.78 TLR8 (0.51) TLR8RAB9AKMT2ACYP1A2HTR3A
SCHEMBL1271431 0.77 CYP1A2 (0.36) TLR8CYP11B2RAB9AKMT2ACYP1A2
SCHEMBL3433191 0.77 TLR8 (0.55) TLR8RAB9A
Phosphine SCHEMBL27716021 0.77 TLR8 (0.52) TLR8RAB9AKMT2ACYP1A2
Hydrochloric Acid SCHEMBL27905861 0.76 TLR8 (0.50) TLR8RAB9AKMT2ACYP1A2HTR3A
SCHEMBL716117 0.76 TSHR (0.50) TLR8HCRTR1HCRTR2CYP1A2HTR3A
Hydrochloric Acid SCHEMBL27476977 0.75 TSHR (0.49) TLR8HCRTR1HCRTR2CYP1A2HTR3A
SCHEMBL28700302 0.74 KDM4E (0.37) MKNK1TLR8HCRTR1HCRTR2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102026985-A Quinazoline derivatives as RAF kinase modulators and methods and uses thereof AMBIT BIOSCIENCES CORPORATON 2011-04-20 CN disclosed