SCHEMBL27846569

SCHEMBL27846569

COc1ccc(-c2ncc(-c3cnc(N4CCN(C)CC4)c(C(F)(F)F)c3)[nH]2)cc1OC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.60
HPGDS O60760 1/20 0.47
NPY5R Q15761 1/20 0.47
MAP4K1 Q92918 6/20 0.47
MEN1 O00255 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
MET P08581 1/20 0.45
IL2 P60568 3/20 0.42
LCK P06239 1/20 0.42
MAP4K3 Q8IVH8 1/20 0.42
TLR9 Q9NR96 2/20 0.42
TLR8 Q9NR97 2/20 0.42
TLR7 Q9NYK1 2/20 0.42
GAK O14976 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
SMPD3 Q9NY59 1/20 0.40
RBP4 P02753 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27863678 0.81 HPGDS (0.58) HPGDSNPY5RMAP4K1MEN1CYP1A2
SCHEMBL532280 0.75 PIK3CA (1.00) PIK3CAMEN1CYP1A2CYP2D6MAPT
SCHEMBL532281 0.73 PIK3CA (0.72) PIK3CAMAP4K1MEN1CYP1A2CYP2D6
SCHEMBL15975825 0.69 PIK3CA (0.89) PIK3CAMEN1CYP1A2CYP2D6MAPT
SCHEMBL16332765 0.68 KCNH2 (0.64) MAP4K1MEN1CYP1A2CYP2D6MAPT
SCHEMBL532219 0.67 PIK3CA (0.82) PIK3CAMEN1KMT2A
SCHEMBL27846714 0.66 HPGDS (0.62) HPGDSNPY5RGAKSMPD3SCN2A
SCHEMBL532220 0.66 PIK3CA (0.59) PIK3CAMAP4K1MEN1CYP1A2KMT2A
SCHEMBL2842992 0.65 HPGDS (1.00) HPGDSNPY5RSMPD3SCN2A
SCHEMBL28976260 0.65 SMN1; SMN2 (0.47) PIK3CAMEN1CYP1A2CYP2D6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102388055-A Imidazo [2, 1-b] [ 1, 3, 4 ] thiadiazole derivatives CT NAC INVESTIGACIONES ONCOLOGICAS CNIO 2012-03-21 CN disclosed