SCHEMBL27847250

SCHEMBL27847250

Cn1cc(-c2cc(Oc3cccc(NC(=O)Nc4ccc(Cl)c(C(F)(F)F)c4)c3)ccn2)cn1

nearest known ligand 0.87

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDR P35968 14/20 0.87
RET P07949 1/20 0.64
CDK8 P49336 2/20 0.59
RAF1 P04049 2/20 0.57
NTRK1 P04629 1/20 0.56
FLT1 P17948 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17179246 0.93 KDR (1.00) KDRRETCDK8RAF1NTRK1
SCHEMBL28793967 0.91 KDR (0.72) KDRRETCDK8NTRK1
SCHEMBL27847472 0.91 KDR (0.72) KDRRETCDK8RAF1NTRK1
SCHEMBL27864410 0.91 KDR (0.72) KDRRETRAF1NTRK1
SCHEMBL5338565 0.90 KDR (0.71) KDRRETRAF1
SCHEMBL27882962 0.90 KDR (0.88) KDRRETRAF1FLT1
SCHEMBL27864336 0.90 KDR (0.71) KDRRETCDK8NTRK1
SCHEMBL27847248 0.90 KDR (0.71) KDRRETRAF1NTRK1
SCHEMBL27846440 0.90 KDR (0.70) KDRRETCDK8RAF1NTRK1
SCHEMBL572529 0.89 KDR (0.85) KDRRETRAF1FLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102408408-A Aryl urea derivative with anti-tumor effect UNIV PEKING FOUNDER GROUP CO 2012-04-11 CN claimed
CN-102408408-A Aryl urea derivative with anti-tumor effect UNIV PEKING FOUNDER GROUP CO 2012-04-11 CN disclosed