SCHEMBL27869740

SCHEMBL27869740

NC(=O)CCCc1ccc2nc(N)nc(C(=O)N3Cc4ccccc4C3)c2c1

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 11/20 0.66
HSP90AB1 P08238 3/20 0.66
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
NAMPT P43490 3/20 0.38
TLR8 Q9NR97 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3076546 0.89 HSP90AA1 (0.69) HSP90AA1HSP90AB1CYP1A2CYP2D6CYP2C19
SCHEMBL3099258 0.89 HSP90AA1 (0.71) HSP90AA1HSP90AB1NAMPT
SCHEMBL12273502 0.88 HSP90AA1 (0.72) HSP90AA1HSP90AB1
SCHEMBL13960641 0.88 HSP90AA1 (0.70) HSP90AA1HSP90AB1
SCHEMBL1768003 0.88 HSP90AA1 (0.66) HSP90AA1HSP90AB1NAMPTTLR8
SCHEMBL16628727 0.87 HSP90AA1 (0.71) HSP90AA1HSP90AB1
SCHEMBL27869741 0.87 HSP90AA1 (0.57) HSP90AA1HSP90AB1NAMPT
SCHEMBL13180105 0.86 HSP90AA1 (0.73) HSP90AA1HSP90AB1NAMPT
SCHEMBL13144772 0.85 HSP90AA1 (0.64) HSP90AA1HSP90AB1CYP1A2CYP2D6CYP2C19
SCHEMBL3086636 0.85 HSP90AA1 (0.64) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102648178-A Quinazoline derivatives MERCK PATENT GMBH 2012-08-22 CN disclosed