SCHEMBL27870231

SCHEMBL27870231

CN1CCN(CCCCOc2cccc([N+](=O)[O-])c2)CC1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.59
PTGS2 P35354 1/20 0.59
HPGD P15428 2/20 0.57
LMNA P02545 1/20 0.57
HRH3 Q9Y5N1 2/20 0.56
CHRNB2 P17787 1/20 0.55
CHRNA4 P43681 1/20 0.55
IKBKB O14920 1/20 0.54
CHRNB4 P30926 1/20 0.54
CHRNA3 P32297 1/20 0.54
DRD3 P35462 1/20 0.52
ALDH1A1 P00352 2/20 0.51
USP2 O75604 1/20 0.51
TSHR P16473 1/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
SIGMAR1 Q99720 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26378399 0.96 LTA4H (0.60) LTA4HPTGS2HPGDLMNAHRH3
SCHEMBL3207509 0.92 LTA4H (0.68) LTA4HPTGS2HPGDLMNAHRH3
SCHEMBL491779 0.89 HRH3 (0.72) LTA4HPTGS2HPGDLMNAHRH3
SCHEMBL5857234 0.88 HRH3 (0.70) LTA4HPTGS2HPGDLMNAHRH3
SCHEMBL27853344 0.86 LTA4H (0.58) LTA4HPTGS2HPGDLMNAHRH3
SCHEMBL18788213 0.86 LTA4H (0.73) LTA4HPTGS2HRH3CHRNB2CHRNA4
SCHEMBL13202242 0.85 LTA4H (0.72) LTA4HPTGS2HRH3CHRNB2CHRNA4
SCHEMBL27853347 0.84 HRH3 (0.78) LTA4HPTGS2HPGDHRH3ALDH1A1
SCHEMBL27870157 0.83 LTA4H (0.49) LTA4HPTGS2HPGDLMNAHRH3
SCHEMBL13949514 0.82 CYP1A2 (0.59) LTA4HPTGS2HRH3CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102464631-B Piperazine substituted 1,3-2-substituted carbamide compounds and the substituted amides compound of piperazine and its production and use 中国科学院上海药物研究所 2016-08-10 CN disclosed
CN-102464631-A Piperazine substituted 1,3-disubstitued urea compounds and piperazine substituted amide compounds, preparation method, and use thereof SHANGHAI INST MATERIA MEDICA 2012-05-23 CN disclosed