SCHEMBL27876232

SCHEMBL27876232

NC(Cc1ccc(-c2cc(OC(c3ccc(F)cc3OC3CCCCC3)C(F)(F)F)ncn2)cc1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TPH1 P17752 19/20 0.48
TPH2 Q8IWU9 10/20 0.48
F2 P00734 1/20 0.43
ESR1 P03372 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
DRD1 P21728 1/20 0.43
PTGS1 P23219 1/20 0.43
SLC6A2 P23975 1/20 0.43
AGTR1 P30556 1/20 0.43
SLC6A4 P31645 1/20 0.43
CCKAR P32238 1/20 0.43
PTGS2 P35354 1/20 0.43
DRD3 P35462 1/20 0.43
SLC6A3 Q01959 1/20 0.43
KMO O15229 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL870506 1.00 TPH1 (0.48) TPH1TPH2F2ESR1ADORA3
SCHEMBL869801 0.99 TPH1 (0.48) TPH1TPH2F2ESR1ADORA3
SCHEMBL27747384 0.99 TPH1 (0.48) TPH1TPH2F2ESR1ADORA3
SCHEMBL27892947 0.92 TPH1 (0.45) TPH1TPH2F2ESR1ADORA3
SCHEMBL869680 0.92 TPH1 (0.50) TPH1TPH2F2ESR1ADORA3
SCHEMBL27726676 0.92 TPH1 (0.46) TPH1TPH2F2ESR1ADORA3
SCHEMBL870039 0.91 TPH1 (0.51) TPH1TPH2F2ESR1ADORA3
SCHEMBL869064 0.89 TPH1 (0.51) TPH1TPH2F2ESR1ADORA3
SCHEMBL27726672 0.89 TPH1 (0.51) TPH1TPH2F2ESR1ADORA3
SCHEMBL27892907 0.89 TPH1 (0.62) TPH1TPH2F2ESR1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102711757-A Methods and assays for treating irritable bowel syndrome LEXICON PHARMACEUTICALS INC 2012-10-03 CN disclosed