SCHEMBL27878769

SCHEMBL27878769

CC(C)n1cc(C#N)c(I)n1

nearest known ligand 0.30

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4361482 0.78 KDM5A (0.33) KDM5AADORA2AADORA1
SCHEMBL24848624 0.77 PIK3CD (0.31) KDM5AADORA2AADORA1
SCHEMBL28239142 0.77 KDM4E (0.32) KDM5AADORA2AADORA1
SCHEMBL8233937 0.77 ADORA2A (0.37) KDM5AADORA2AADORA1
SCHEMBL26161133 0.74 ADORA2A (0.32) KDM5AADORA2AADORA1
SCHEMBL21802995 0.74
SCHEMBL15723768 0.73 LRRK2 (0.36) KDM5A
SCHEMBL22574524 0.71 ADORA2A (0.41) ADORA2AADORA1
SCHEMBL15808415 0.67 HTT (0.36)
SCHEMBL15703081 0.67 ADORA2A (0.31) ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104744491-B Benzo oxazepine * PI3K inhibitor compounds and application method 霍夫曼-拉罗奇有限公司 2017-07-11 CN disclosed
CN-102762576-A Benzoxazepine PI3K inhibitor compounds and methods of use HOFFMANN LA ROCHE 2012-10-31 CN disclosed