SCHEMBL28239142

SCHEMBL28239142

CC(C)n1cc(C#N)c(Br)n1

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
KDM5A P29375 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30
AR P10275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4361482 0.78 KDM5A (0.33) KDM4EALDH1A1KDM5AADORA2AADORA1
SCHEMBL8233937 0.77 ADORA2A (0.37) KDM4EALDH1A1KDM5AADORA2AADORA1
SCHEMBL24848624 0.77 PIK3CD (0.31) KDM5AADORA2AADORA1
SCHEMBL27878769 0.77 KDM5A (0.30) KDM5AADORA2AADORA1
SCHEMBL26161133 0.74 ADORA2A (0.32) KDM5AADORA2AADORA1
SCHEMBL16654819 0.74
SCHEMBL15723770 0.73 KDM5A (0.34) KDM5AADORA2AADORA1
SCHEMBL15723768 0.73 LRRK2 (0.36) ALDH1A1SMN1; SMN2KDM5AAR
SCHEMBL28932516 0.69 ADORA2A (0.40) ADORA2AADORA1
SCHEMBL15808415 0.67 HTT (0.36) KDM4EALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108530436-A A kind of pyrazole compound and its preparation method and application 黄传满 2018-09-14 CN disclosed