SCHEMBL27880337

SCHEMBL27880337

CCCCCN(C(N)=O)c1ncc2ccccc2n1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 7/20 0.42
TLR8 Q9NR97 4/20 0.42
NPC1 O15118 1/20 0.41
JAK2 O60674 1/20 0.41
RAB9A P51151 1/20 0.41
PAX8 Q06710 1/20 0.41
ELANE P08246 1/20 0.40
PTPN11 Q06124 1/20 0.40
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17941675 0.84 TLR8 (0.39) TRPV1TLR8NPC1JAK2RAB9A
SCHEMBL11769407 0.80 TLR8 (0.46) TRPV1TLR8ELANE
SCHEMBL4763663 0.79 NPC1 (0.42) NPC1JAK2RAB9APAX8ALDH1A1
SCHEMBL3055011 0.73 NPC1 (0.65) NPC1JAK2RAB9APAX8ALDH1A1
SCHEMBL11635003 0.73 SPHK2 (0.50) NPC1RAB9AALDH1A1
SCHEMBL28221454 0.73 TRPV1 (0.35) TRPV1RAB9APTPN11
SCHEMBL6424475 0.72 NPC1 (0.68) NPC1JAK2RAB9APAX8ALDH1A1
SCHEMBL1082836 0.72 NPC1 (0.68) NPC1JAK2RAB9APAX8ALDH1A1
SCHEMBL11344801 0.72 NPC1 (0.68) NPC1JAK2RAB9APAX8ALDH1A1
SCHEMBL7096422 0.72 NPC1 (0.68) NPC1JAK2RAB9APAX8ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104292170-A Quinazolinyl-aryl urea derivatives with antitumor function and application thereof UNIV GUANGXI NORMAL 2015-01-21 CN disclosed
CN-104292170-A Quinazolinyl-aryl urea derivatives with antitumor function and application thereof UNIV GUANGXI NORMAL 2015-01-21 CN disclosed
CN-102532103-B Quinazolinyl aryl urea derivatives and preparation method and application thereof TIANJIN INST PHARM RESEARCH 2014-07-09 CN disclosed
CN-102532103-B Quinazolinyl aryl urea derivatives and preparation method and application thereof TIANJIN INST PHARM RESEARCH 2014-07-09 CN disclosed
CN-102532103-A Quinazolinyl aryl urea derivatives and preparation method and application thereof TIANJIN INST PHARM RESEARCH 2012-07-04 CN disclosed
CN-102532103-A Quinazolinyl aryl urea derivatives and preparation method and application thereof TIANJIN INST PHARM RESEARCH 2012-07-04 CN disclosed