SCHEMBL27883183

SCHEMBL27883183

Cc1cc(C)nc(N2CC3CN(C(=O)c4c(Cl)cccc4CN)CC3C2)n1

nearest known ligand 0.75

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 20/20 0.75
HCRTR2 O43614 20/20 0.75
KCNH2 Q12809 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1671072 0.86 HCRTR1 (1.00) HCRTR1HCRTR2KCNH2
SCHEMBL27900616 0.80 HCRTR1 (0.74) HCRTR1HCRTR2
SCHEMBL1672522 0.80 HCRTR1 (1.00) HCRTR1HCRTR2KCNH2
SCHEMBL1671303 0.78 HCRTR1 (1.00) HCRTR1HCRTR2
SCHEMBL27900618 0.76 HCRTR1 (0.74) HCRTR1HCRTR2
SCHEMBL1671476 0.76 HCRTR1 (1.00) HCRTR1HCRTR2
SCHEMBL1671620 0.76 HCRTR1 (1.00) HCRTR1HCRTR2
SCHEMBL1671991 0.75 HCRTR1 (1.00) HCRTR1HCRTR2
SCHEMBL27883254 0.75 HCRTR1 (0.75) HCRTR1HCRTR2KCNH2
SCHEMBL6923525 0.74 HCRTR1 (1.00) HCRTR1HCRTR2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102781942-A Disubstituted octahy-dropyrrolo [3,4-c]pyrroles as orexin receptor modulators JANSSEN PHARMACEUTICA NV 2012-11-14 CN claimed