SCHEMBL2789205

SCHEMBL2789205

Cc1ccc2cc(-c3cccnc3)[nH]c2c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.68
MAP2K4 P45985 1/20 0.51
ITK Q08881 4/20 0.51
CYP2A6 P11509 3/20 0.50
NPY5R Q15761 2/20 0.49
KDM4E B2RXH2 3/20 0.46
HSD17B10 Q99714 3/20 0.46
NPC1 O15118 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
CYP3A4 P08684 2/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7946248 0.88 CYP19A1 (0.68) CYP19A1MAP2K4ITKCYP2A6NPY5R
SCHEMBL1606072 0.83 CYP19A1 (0.65) CYP19A1MAP2K4CYP2A6NPY5RNPC1
SCHEMBL1605712 0.82 CYP19A1 (0.68) CYP19A1CYP2A6NPY5RHPGDCYP3A4
SCHEMBL1605273 0.82 CYP19A1 (0.68) CYP19A1CYP2A6NPY5RKDM4ENPC1
SCHEMBL1120933 0.81 CYP19A1 (0.62) CYP19A1ITKNPY5RKDM4EHSD17B10
SCHEMBL29790209 0.81 CYP19A1 (1.00) CYP19A1ITKKDM4EHSD17B10NPC1
SCHEMBL2789486 0.81 CYP19A1 (1.00) CYP19A1ITKKDM4EHSD17B10NPC1
SCHEMBL13541758 0.80 RAB9A (0.63) CYP19A1ITKKDM4EHSD17B10NPC1
Hydrochloric Acid SCHEMBL27830550 0.80 CYP19A1 (0.97) CYP19A1ITKKDM4EHSD17B10NPC1
SCHEMBL4568283 0.78 CYP19A1 (0.58) CYP19A1CYP2A6NPY5RKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed