SCHEMBL278926

SCHEMBL278926

C=C(/N=C/c1cc(Cl)ccc1O[C@H]1CC[C@@H](O[Si](C)(C)C(C)(C)C)CC1)O[Si](C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.37
TSHR P16473 2/20 0.37
CNR2 P34972 1/20 0.33
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
FPR2 P25090 1/20 0.31
PROKR1 Q8TCW9 1/20 0.31
RBP4 P02753 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL279050 1.00 HPGD (0.37) HPGDTSHRCNR2MEN1KMT2A
SCHEMBL279490 0.85 HPGD (0.36) HPGDTSHR
SCHEMBL274631 0.85 HPGD (0.36) HPGDTSHR
SCHEMBL278931 0.84 CHEK1 (0.38) HPGDTSHRCNR2
SCHEMBL275247 0.84 CHEK1 (0.38) HPGDTSHRCNR2
SCHEMBL279174 0.83 HPGD (0.38) HPGDTSHRCNR2MEN1KMT2A
SCHEMBL274636 0.83 HPGD (0.38) HPGDTSHRCNR2MEN1KMT2A
SCHEMBL275642 0.83 HPGD (0.40) HPGDTSHRMEN1KMT2A
SCHEMBL278953 0.83 HPGD (0.40) HPGDTSHRMEN1KMT2A
SCHEMBL279042 0.80 CACNB4 (0.37) HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8134001-B2 Spiroindolinone derivatives HOFFMANN-LA ROCHE INC. (US) 2012-03-13 US disclosed
US-20090156610-A1 Spiroindolinone Derivatives DING QINGJIE 2009-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156610-A1 Spiroindolinone Derivatives SDHA, AR, XPOT HPGD 482/4885TSHR 1261/4885CNR2 4264/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.