SCHEMBL27892829

SCHEMBL27892829

COc1c(Cl)cncc1-c1cccc(F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 3/20 0.47
CSNK1D P48730 3/20 0.46
GSK3A P49840 3/20 0.46
GSK3B P49841 3/20 0.46
DYRK1A Q13627 3/20 0.46
AURKB Q96GD4 3/20 0.46
RPS6KB1 P23443 2/20 0.46
NTRK2 Q16620 1/20 0.46
SLC22A12 Q96S37 1/20 0.46
MAPK10 P53779 1/20 0.44
PDGFRB P09619 1/20 0.43
PDGFRA P16234 1/20 0.43
RPS6KA3 P51812 2/20 0.41
PLK4 O00444 2/20 0.41
AURKA O14965 2/20 0.41
DAPK3 O43293 2/20 0.41
CHEK2 O96017 2/20 0.41
CDK1 P06493 2/20 0.41
PIM1 P11309 2/20 0.41
CDK2 P24941 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27892837 0.86 FYN (0.48) FYNCSNK1DGSK3AGSK3BDYRK1A
SCHEMBL27892827 0.85 FYN (0.53) FYNCSNK1DGSK3AGSK3BDYRK1A
SCHEMBL27876162 0.81 RPS6KA3 (0.44) FYNMAPK10RPS6KA3BRAFCYP11B2
SCHEMBL16297083 0.75 CYP1A1 (0.51) FYNRPS6KB1MAPK10CYP11B2MAPK1
SCHEMBL1770160 0.75 CSNK1D (0.43) FYNCSNK1DGSK3AGSK3BDYRK1A
SCHEMBL11178949 0.74 CSNK1D (0.48) CSNK1DGSK3AGSK3BDYRK1AAURKB
SCHEMBL27876161 0.74 PDE4B (0.56) FYNCSNK1DGSK3AGSK3BDYRK1A
SCHEMBL27876164 0.73 DHPS (0.40) BRAFCYP11B2IDO1CYP11B1
SCHEMBL8220816 0.72 FYN (0.45) FYNPDGFRBPDGFRAMAPK1KIT
SCHEMBL15011871 0.72 CYP1A1 (0.47) RPS6KB1MAPK10CYP11B2MAPK1PRKAA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102712589-A Aryl-pyridine derivatives as aldosterone synthase inhibitors NOVARTIS AG 2012-10-03 CN claimed
CN-102712589-A Aryl-pyridine derivatives as aldosterone synthase inhibitors NOVARTIS AG 2012-10-03 CN disclosed