SCHEMBL278977

SCHEMBL278977

C=C(/N=C/c1cc(I)ccc1OC1CCOCC1)O[Si](C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.36
PDE4D Q08499 9/20 0.34
PDE4B Q07343 6/20 0.34
PDE4A P27815 5/20 0.34
PDE4C Q08493 5/20 0.34
KAT2B Q92831 1/20 0.34
BAZ2B Q9UIF8 1/20 0.34
QPCT Q16769 1/20 0.32
QPCTL Q9NXS2 1/20 0.32
IKBKE Q14164 5/20 0.31
TBK1 Q9UHD2 5/20 0.31
CHEK1 O14757 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL276886 1.00 SYK (0.36) SYKPDE4DPDE4BPDE4APDE4C
SCHEMBL276159 0.90 PDE4D (0.35) PDE4DPDE4BPDE4APDE4C
SCHEMBL279509 0.90 PDE4D (0.35) PDE4DPDE4BPDE4APDE4C
SCHEMBL275247 0.87 CHEK1 (0.38) SYKPDE4DPDE4BPDE4APDE4C
SCHEMBL278978 0.87 SYK (0.36) SYKPDE4DPDE4BPDE4APDE4C
SCHEMBL276376 0.87 SYK (0.39) SYKPDE4DPDE4BPDE4APDE4C
SCHEMBL278931 0.87 CHEK1 (0.38) SYKPDE4DPDE4BPDE4APDE4C
SCHEMBL279161 0.87 SYK (0.39) SYKPDE4DPDE4BPDE4APDE4C
SCHEMBL7790693 0.85 PDE4D (0.35) SYKPDE4DPDE4BPDE4APDE4C
SCHEMBL279337 0.80 PDE4B (0.44) PDE4DPDE4BPDE4APDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8134001-B2 Spiroindolinone derivatives HOFFMANN-LA ROCHE INC. (US) 2012-03-13 US disclosed
US-20090156610-A1 Spiroindolinone Derivatives DING QINGJIE 2009-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156610-A1 Spiroindolinone Derivatives SDHA, AR, XPOT SYK 2511/4885PDE4D 2759/4885PDE4B 3594/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.