SCHEMBL2789976

SCHEMBL2789976

COc1cccc(CN(C(=O)C2CNCC[C@@H]2NC(=O)c2ccc(OCCOc3c(Cl)cc(C)cc3Cl)cc2)C2CC2)c1C

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
REN P00797 20/20 0.67
CYP3A4 P08684 13/20 0.67
KCNH2 Q12809 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL695697 0.99 REN (0.66) RENCYP3A4KCNH2
SCHEMBL2792552 0.95 REN (0.63) RENCYP3A4KCNH2
Hydrochloric Acid SCHEMBL695392 0.94 REN (0.62) RENCYP3A4KCNH2
Hydrochloric Acid SCHEMBL696345 0.94 REN (0.62) RENCYP3A4KCNH2
SCHEMBL2788513 0.93 REN (0.77) RENCYP3A4
SCHEMBL694821 0.93 REN (0.77) RENCYP3A4
Hydrochloric Acid SCHEMBL694530 0.92 REN (0.76) RENCYP3A4
Hydrochloric Acid SCHEMBL2691553 0.92 REN (0.76) RENCYP3A4
Hydrochloric Acid SCHEMBL695376 0.92 REN (0.76) RENCYP3A4
SCHEMBL695702 0.91 REN (0.73) RENCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010122580-A2 NOVEL COMPOUNDS AS INHIBITORS OF RENIN CADILA HEALTHCARE LIMITED (IN) 2010-10-28 WO claimed