SCHEMBL27900600

SCHEMBL27900600

Cc1ccnc(-c2ccc(F)cc2C(=O)c2cc(F)ccc2-c2cc(C)ccn2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 9/20 0.58
HCRTR2 O43614 9/20 0.58
ABL1 P00519 1/20 0.47
BCR P11274 1/20 0.47
CCR1 P32246 1/20 0.47
CCR5 P51681 1/20 0.47
CCR8 P51685 1/20 0.47
TACR3 P29371 1/20 0.44
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
TP53 P04637 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KDM1A O60341 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
KMO O15229 1/20 0.40
NFKB1 P19838 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27900620 0.88 HCRTR1 (0.56) HCRTR1HCRTR2ABL1BCRCCR1
SCHEMBL10014733 0.81 HCRTR1 (0.45) HCRTR1HCRTR2ABL1BCRCCR1
SCHEMBL29766750 0.79 CCR1 (0.55) HCRTR1HCRTR2ABL1BCRCCR1
SCHEMBL16910413 0.79 CCR1 (0.55) HCRTR1HCRTR2ABL1BCRCCR1
SCHEMBL503953 0.79 CCR1 (0.55) HCRTR1HCRTR2ABL1BCRCCR1
SCHEMBL28802210 0.79 HCRTR1 (0.57) HCRTR1HCRTR2CCR1CCR5CCR8
SCHEMBL27870875 0.78 HCRTR1 (0.54) HCRTR1HCRTR2CCR1CCR5CCR8
SCHEMBL27854353 0.77 NPC1 (0.45) HCRTR1HCRTR2NPC1RAB9AKMO
SCHEMBL6924236 0.76 HCRTR1 (1.00) HCRTR1HCRTR2
SCHEMBL6130738 0.75 CCR1 (0.50) HCRTR1HCRTR2ABL1BCRCCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102781942-A Disubstituted octahy-dropyrrolo [3,4-c]pyrroles as orexin receptor modulators JANSSEN PHARMACEUTICA NV 2012-11-14 CN claimed
CN-102781942-A Disubstituted octahy-dropyrrolo [3,4-c]pyrroles as orexin receptor modulators JANSSEN PHARMACEUTICA NV 2012-11-14 CN disclosed