SCHEMBL27907249

SCHEMBL27907249

CN(C)Cc1ccc(N(C)c2cc(N)ncn2)cc1C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.37
CYP2D6 P10635 2/20 0.37
CA2 P00918 1/20 0.35
CHKA P35790 1/20 0.35
SLC6A2 P23975 4/20 0.34
SLC6A4 P31645 4/20 0.34
SLC6A3 Q01959 3/20 0.34
POLQ O75417 3/20 0.33
CYP3A4 P08684 2/20 0.32
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
ALOX15 P16050 1/20 0.32
CYP2C19 P33261 1/20 0.32
HCK P08631 1/20 0.32
NR2C2 P49116 1/20 0.32
AAK1 Q2M2I8 1/20 0.32
EGFR P00533 1/20 0.31
CD274 Q9NZQ7 1/20 0.30
JAK2 O60674 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL374483 0.78 CDK5 (0.46) CYP1A2CYP2D6CA2CHKACYP3A4
SCHEMBL374610 0.71 NR1H2 (0.51) CYP1A2CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL30401867 0.71 NR1H2 (0.51) CYP1A2CYP2D6SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL16054675 0.70 NR1H2 (0.50) CYP1A2CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL27907260 0.69 ALDH1A1 (0.46) CA2CHKACYP3A4ALDH1A1LMNA
SCHEMBL27907258 0.67 EGFR (0.44) ALDH1A1EGFR
SCHEMBL374500 0.67 CYP1A2 (0.47) CYP1A2CYP2D6CYP3A4ALDH1A1LMNA
SCHEMBL13960088 0.66 SLC6A4 (0.46) CYP1A2CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL7780176 0.65 NR3C2 (0.36) CYP2D6CYP3A4
SCHEMBL24399683 0.65 SLC6A4 (0.52) CYP1A2CYP2D6SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103121973-A Pyrimidine urea derivatives as kinase inhibitors NOVARTIS AG 2013-05-29 CN disclosed
CN-103121972-A Pyrimidine urea derivatives as kinase inhibitors NOVARTIS AG 2013-05-29 CN disclosed