SCHEMBL27908484

SCHEMBL27908484

CC(=O)Oc1coc(C2CCCN2C(=O)OCc2ccccc2)n1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AADAT Q8N5Z0 2/20 0.51
ACE2 Q9BYF1 3/20 0.46
CTSK P43235 2/20 0.46
PREP P48147 3/20 0.46
TMEM97 Q5BJF2 2/20 0.45
SIGMAR1 Q99720 2/20 0.45
HSD17B10 Q99714 1/20 0.44
CTSB P07858 1/20 0.43
CTSS P25774 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27891373 1.00 AADAT (0.51) AADATACE2CTSKPREPTMEM97
SCHEMBL953139 0.86 AADAT (0.52) AADATACE2PREPTMEM97SIGMAR1
SCHEMBL953138 0.86 AADAT (0.52) AADATACE2PREPTMEM97SIGMAR1
SCHEMBL18850754 0.84 HCRTR1 (0.53) AADATACE2PREPTMEM97SIGMAR1
SCHEMBL475407 0.82 AADAT (0.51) AADATACE2CTSKPREPTMEM97
SCHEMBL475406 0.82 AADAT (0.51) AADATACE2CTSKPREPTMEM97
SCHEMBL27891374 0.82 AADAT (0.49) AADATACE2PREPTMEM97SIGMAR1
SCHEMBL952909 0.78 PREP (0.50) AADATACE2PREPTMEM97SIGMAR1
SCHEMBL952907 0.78 PREP (0.50) AADATACE2PREPTMEM97SIGMAR1
SCHEMBL4220121 0.77 PREP (0.50) AADATACE2PREPTMEM97SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101868457-B (3-hydroxy-4-amino-but-2-yl) -3- (2-thiazol-2-yl-pyrrolidine-1-carbonyl) benzamide derivatives and related compounds as beta-secretase inhibitors for use in therapy COMENTIS INC 2013-02-13 CN disclosed