SCHEMBL27913072

SCHEMBL27913072

CC(C)(C)C(=O)OC(C)(C)c1cc(Cc2ccc(Cl)cc2)nc(NC2CCNCC2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK4 O00444 1/20 0.42
PAK4 O96013 1/20 0.42
PSEN1 P49768 4/20 0.42
PSEN2 P49810 4/20 0.42
APH1B Q8WW43 4/20 0.42
NCSTN Q92542 4/20 0.42
APH1A Q96BI3 4/20 0.42
PSENEN Q9NZ42 4/20 0.42
IKBKB O14920 1/20 0.38
SSTR4 P31391 2/20 0.37
SSTR1 P30872 1/20 0.37
HRH1 P35367 2/20 0.36
DDR1 Q08345 2/20 0.35
CDK2 P24941 3/20 0.34
CDK9 P50750 2/20 0.34
HRH4 Q9H3N8 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
LCK P06239 1/20 0.34
ITK Q08881 1/20 0.34
AURKB Q96GD4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2269500 0.85 PSEN1 (0.54) PLK4PAK4PSEN1PSEN2APH1B
Tert-Butyl Formate SCHEMBL27913074 0.81 PSEN1 (0.47) PLK4PAK4PSEN1PSEN2APH1B
SCHEMBL2270043 0.74 PSEN1 (0.51) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL12078284 0.71 PSEN1 (0.48) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL12078283 0.71 PSEN1 (0.48) PSEN1PSEN2APH1BNCSTNAPH1A
Hydrochloric Acid SCHEMBL12078705 0.71 PSEN1 (0.51) PLK4PAK4PSEN1PSEN2APH1B
SCHEMBL2354610 0.69 ALDH1A1 (0.50)
SCHEMBL27689356 0.67 DDR1 (0.50) SSTR4SSTR1DDR1
SCHEMBL2271410 0.67 PSEN1 (0.51) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2278329 0.66 PSEN1 (0.77) PLK4PAK4PSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103025724-A Piperidine derivatives HOFFMANN LA ROCHE 2013-04-03 CN disclosed