SCHEMBL27923391

SCHEMBL27923391

Nc1ccc2ncnc(Nc3ccc(F)cc3)c2c1

nearest known ligand 0.73

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EGFR P00533 16/20 0.73
MEN1 O00255 1/20 0.61
USP2 O75604 1/20 0.61
ALDH1A1 P00352 1/20 0.61
LMNA P02545 1/20 0.61
CYP1A2 P05177 1/20 0.61
CYP3A4 P08684 1/20 0.61
CYP2D6 P10635 1/20 0.61
TSHR P16473 1/20 0.61
CYP2C19 P33261 1/20 0.61
KMT2A Q03164 1/20 0.61
HIF1A Q16665 1/20 0.61
CLK4 Q9HAZ1 1/20 0.61
ERBB2 P04626 3/20 0.60
CD38 P28907 1/20 0.60
RAF1 P04049 1/20 0.59
BRAF P15056 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2103341 0.91 EGFR (0.82) EGFRMEN1ALDH1A1LMNAKMT2A
SCHEMBL27878333 0.89 USP2 (0.65) EGFRMEN1USP2ALDH1A1LMNA
SCHEMBL28086820 0.88 EGFR (0.73) EGFRMEN1USP2ALDH1A1LMNA
SCHEMBL4586685 0.86 EGFR (0.75) EGFRMEN1ALDH1A1LMNAKMT2A
SCHEMBL27685863 0.85 EGFR (0.73) EGFRLMNAERBB2CD38
SCHEMBL30513 0.84 EGFR (1.00) EGFRLMNACYP1A2CYP3A4HIF1A
SCHEMBL29690398 0.84 EGFR (1.00) EGFRLMNACYP1A2CYP3A4HIF1A
Hydrochloric Acid SCHEMBL7760887 0.84 EGFR (0.76) EGFRERBB2
SCHEMBL28475211 0.84 CD38 (0.62) EGFRMEN1USP2ALDH1A1LMNA
SCHEMBL5568874 0.84 HTT (0.74) EGFRMEN1USP2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103382182-B Phenylurea coupling quinazoline compounds and preparation method thereof, pharmaceutical composition and medicinal usage 河北医科大学 2016-08-10 CN disclosed
CN-105753793-A Aroylurea coupled quinazoline type compound and preparation method, pharmaceutical composition and pharmaceutical uses thereof 河北医科大学 2016-07-13 CN disclosed
CN-103382182-A Phenylurea coupling quinazoline compound, and preparation method, pharmaceutical composition and pharmaceutical use thereof UNIV HEBEI MEDICAL 2013-11-06 CN disclosed