SCHEMBL27923799

SCHEMBL27923799

NCc1ccccc1P(C1CCCCC1)C1CCCCC1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
OPRL1 P41146 1/20 0.37
PNMT P11086 3/20 0.35
DPP4 P27487 2/20 0.33
BRD4 O60885 1/20 0.33
CARM1 Q86X55 2/20 0.32
PRMT1 Q99873 2/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
AOC3 Q16853 5/20 0.32
AOC1 P19801 4/20 0.32
NCF1 P14598 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1315359 0.80 ROCK2 (0.35)
SCHEMBL16694657 0.80 KMT2A (0.39) CYP2D6
SCHEMBL1314189 0.78 ROCK2 (0.33)
SCHEMBL17583591 0.77 ROCK2 (0.33)
SCHEMBL28859669 0.76 KMT2A (0.31)
SCHEMBL14905782 0.76 GAA (0.43) CYP3A4
SCHEMBL520084 0.75 BCHE (0.37)
SCHEMBL2846316 0.75 TAAR1 (0.34) CYP3A4CYP2D6
SCHEMBL16695057 0.75 KMT2A (0.35)
Formaldehyde SCHEMBL17583570 0.73 ROCK2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103384665-B The method for preparing gyrase and topoisomerase enzyme inhibitor 斯派罗吹耐姆公司 2018-01-09 CN disclosed
CN-103384665-A Process of making gyrase and topoisomerase IV inhibitors VERTEX PHARMA 2013-11-06 CN disclosed