SCHEMBL27924985

SCHEMBL27924985

CC(c1ccc(-c2nn(C)cc2-c2ccncc2)nc1)[Si](C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CSNK1D P48730 2/20 0.47
MAPK14 Q16539 2/20 0.47
MAPK13 O15264 1/20 0.47
CSNK1E P49674 1/20 0.47
MAPK12 P53778 1/20 0.47
MAPK11 Q15759 1/20 0.47
BRAF P15056 13/20 0.46
MAPK3 P27361 4/20 0.43
MAPK1 P28482 4/20 0.43
PDE10A Q9Y233 4/20 0.40
MAP4K4 O95819 1/20 0.38
EGFR P00533 1/20 0.38
FRK P42685 1/20 0.38
MAPK9 P45984 1/20 0.38
CSNK1A1 P48729 1/20 0.38
LGALS3 P17931 1/20 0.37
PDE4D Q08499 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15022322 0.78 CSNK1D (0.52) CSNK1DMAPK14MAPK13CSNK1EMAPK12
SCHEMBL15022080 0.75 PDE10A (0.49) CSNK1DMAPK14MAPK13CSNK1EMAPK12
SCHEMBL27924982 0.75 MAPK13 (0.46) CSNK1DMAPK14MAPK13CSNK1EMAPK12
SCHEMBL15022065 0.75 PDE10A (0.49) CSNK1DMAPK14MAPK13CSNK1EMAPK12
SCHEMBL27907019 0.73 MAPK14 (0.56) CSNK1DMAPK14MAPK13CSNK1EMAPK12
SCHEMBL15022316 0.67 MAPK13 (0.62) CSNK1DMAPK14MAPK13CSNK1EMAPK12
SCHEMBL5258671 0.67 MAPK13 (0.71) CSNK1DMAPK14MAPK13CSNK1EMAPK12
SCHEMBL27924978 0.66 MAPK13 (0.61) CSNK1DMAPK14MAPK13CSNK1EMAPK12
SCHEMBL15023023 0.66 PDE10A (0.52) PDE10ALGALS3PDE4D
SCHEMBL5258392 0.66 MAPK13 (0.74) CSNK1DMAPK14MAPK13CSNK1EMAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103159738-B The heteroaryl aroma compounds of alkynyl bridging and application thereof 上海泓博智源医药股份有限公司 2016-09-07 CN disclosed
CN-103159738-A Mixed aromatic compound of alkynyl bridging and application thereof SHANGHAI HONGBO ZHIYUAN MEDICAL TECHNOLOGY CO LTD 2013-06-19 CN disclosed