Losoxantrone

Losoxantrone

SCHEMBL27927741

O=C1c2c(O)cccc2-c2nn(CCNCCO)c3ccc(NCCNCCO)c1c23.[CH2]C

nearest known ligand 0.94

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 11/20 0.94
MEN1 O00255 3/20 0.48
USP2 O75604 3/20 0.48
LMNA P02545 3/20 0.48
RECQL P46063 3/20 0.48
KMT2A Q03164 3/20 0.48
TP53 P04637 2/20 0.48
MAPK1 P28482 2/20 0.48
BLM P54132 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
TDP1 Q9NUW8 2/20 0.48
NSD2 O96028 2/20 0.48
CSNK2A1 P68400 2/20 0.48
HTT P42858 2/20 0.48
NPC1 O15118 1/20 0.48
SLC22A2 O15244 1/20 0.48
SLC22A1 O15245 1/20 0.48
CACNA1F O60840 1/20 0.48
SLC22A3 O75751 1/20 0.48
EGFR P00533 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Losoxantrone SCHEMBL61319 0.97 TOP2A (1.00) TOP2AMEN1USP2LMNARECQL
Losoxantrone SCHEMBL29360703 0.97 TOP2A (1.00) TOP2AMEN1USP2LMNARECQL
Losoxantrone SCHEMBL6685621 0.96 TOP2A (0.98) TOP2AMEN1USP2LMNARECQL
Losoxantrone SCHEMBL29409658 0.96 TOP2A (0.98) TOP2AMEN1USP2LMNARECQL
Losoxantrone SCHEMBL5170 0.95 TOP2A (0.96) TOP2AMEN1USP2LMNARECQL
SCHEMBL10800466 0.94 TOP2A (0.90) TOP2AMEN1USP2LMNARECQL
Losoxantrone SCHEMBL27975856 0.93 TOP2A (0.88) TOP2AMEN1USP2LMNARECQL
SCHEMBL22877226 0.91 TOP2A (0.87) TOP2AMEN1USP2LMNARECQL
SCHEMBL18689529 0.91 TOP2A (0.87) TOP2AMEN1USP2LMNARECQL
SCHEMBL10805434 0.90 TOP2A (0.86) TOP2AMEN1USP2LMNARECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102892779-B Neuregulin antagonist and the purposes in treatment cancer thereof 基因泰克公司 2016-12-21 CN disclosed
CN-102580084-B The fixed dosage of HER antibody is administered 健泰科生物技术公司 2016-11-23 CN disclosed
CN-106148547-A Diagnostic method and composition for treatment of cancer 霍夫曼-拉罗奇有限公司 2016-11-23 CN disclosed
CN-104011078-B Anti-poly-ubiquitin antibody and using method 健泰科生物技术公司 2016-11-09 CN disclosed
CN-103596983-B Anti-FGFR4 antibody and using method 霍夫曼-拉罗奇有限公司 2016-10-26 CN disclosed
CN-102770158-B Antibody formulations 霍夫曼-拉罗奇有限公司 2016-10-19 CN disclosed
CN-103554263-B Apoptotic anti-IgE antibodies in conjunction with the IgE that film combines 健泰科生物技术公司 2016-09-28 CN disclosed
CN-103030696-B Antibody and immune conjugate and application thereof 健泰科生物技术公司 2016-09-28 CN disclosed
CN-103649117-B Fc variant and the method for generation thereof 霍夫曼-拉罗奇有限公司 2016-09-14 CN disclosed
CN-103396485-B The method and composition of targeting polyubiquitin 健泰科生物技术公司 2016-08-10 CN disclosed
CN-105793288-A Anti-PDL1 antibody formulations 豪夫迈·罗氏有限公司 2016-07-20 CN disclosed
CN-105744954-A anti-RSPO 2 and/or anti-RSPO 3 antibodies and uses thereof 豪夫迈·罗氏有限公司 2016-07-06 CN disclosed
CN-103304667-A Humanized anti-beta7 antagonists and uses therefor GENENTECH INC 2013-09-18 CN disclosed
CN-101094868-B Humanized anti-beta 7 antagonists and uses thereof GENENTECH INC 2013-07-10 CN disclosed