SCHEMBL27934296

SCHEMBL27934296

O=C(NC1CCOCC1)c1cncnc1C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 3/20 0.45
HDAC6 Q9UBN7 2/20 0.44
HDAC4 P56524 1/20 0.44
TRPV1 Q8NER1 2/20 0.42
IRAK4 Q9NWZ3 2/20 0.41
WDR5 P61964 1/20 0.41
CSNK2A2 P19784 1/20 0.41
CSNK2A1 P68400 1/20 0.41
CNR2 P34972 3/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C19 P33261 2/20 0.40
CYP1A2 P05177 1/20 0.40
GABRA5 P31644 1/20 0.40
SCN9A Q15858 1/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
PIM1 P11309 1/20 0.39
PIK3C3 Q8NEB9 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25420116 0.81 CNR2 (0.59) CNR2CYP2D6CYP2C19CYP1A2CYP3A4
SCHEMBL5099923 0.77 GAA (0.50) PDE4BHDAC6HDAC4TRPV1CSNK2A2
SCHEMBL6451201 0.72 CNR2 (0.53) HDAC6HDAC4CNR2CYP2D6CYP2C19
SCHEMBL16879004 0.71 PIM1 (0.45) PDE4BIRAK4CSNK2A2CSNK2A1PIM1
SCHEMBL13503354 0.70 CNR2 (0.62) CNR2CYP2D6CYP2C19CYP1A2CYP3A4
SCHEMBL20337733 0.70 WDR5 (0.44) IRAK4WDR5
SCHEMBL13503355 0.70 CNR2 (0.61) CNR2CYP2D6CYP2C19CYP1A2CYP3A4
SCHEMBL13503356 0.70 CNR2 (0.76) CNR2CYP2D6CYP2C19CYP1A2CYP3A4
SCHEMBL13503327 0.70 CNR2 (0.76) CNR2CYP2D6CYP2C19CYP1A2CYP3A4
SCHEMBL13503361 0.70 CNR2 (0.76) CNR2CYP2D6CYP2C19CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103265517-A 3-substituted coumarin derivative and use thereof UNIV ZHEJIANG 2013-08-28 CN disclosed