SCHEMBL27934814

SCHEMBL27934814

CC(C)(C)OC(=O)NCCCCN1CCN(c2nc(C(N)=O)c(OCc3ccccc3)c3ncccc23)CC1

nearest known ligand 0.50

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.50
SIGMAR1 Q99720 2/20 0.45
DRD3 P35462 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10012640 0.94 DRD2 (0.51) DRD2SIGMAR1DRD3
SCHEMBL1654652 0.93 DRD2 (0.52) DRD2SIGMAR1DRD3
SCHEMBL10012965 0.84 DRD2 (0.43) DRD2SIGMAR1DRD3
SCHEMBL10011586 0.81 DRD2 (0.41) DRD2DRD3
SCHEMBL27935081 0.81 CYP3A4 (0.46)
SCHEMBL12781936 0.80 DRD2 (0.41) DRD2SIGMAR1DRD3
SCHEMBL27949680 0.77 CYP3A4 (0.41)
SCHEMBL1654200 0.75 CYP3A4 (0.47)
SCHEMBL10013000 0.74 CYP3A4 (0.46)
SCHEMBL17861451 0.73 DRD2 (0.60) DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103459390-A Macrocyclic integrase inhibitors for use in the treatment of feline immunodeficiency virus ELANCO ANIMAL HEALTH IRELAND 2013-12-18 CN disclosed