Nolatrexed

Nolatrexed

SCHEMBL27935384

Cc1ccc2nc(N)[nH]c(=O)c2c1Sc1ccncc1.Cl

nearest known ligand 0.97

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

TYMS

The experimentally established mechanism targets of Nolatrexed. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TYMS known ✓ P04818 20/20 0.97
DHFR P00374 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nolatrexed SCHEMBL29420099 1.00 TYMS (0.97) TYMSDHFR
Nolatrexed SCHEMBL316632 1.00 TYMS (0.97) TYMSDHFR
Nolatrexed SCHEMBL710461 0.99 TYMS (1.00) TYMSDHFR
SCHEMBL7826662 0.86 TYMS (1.00) TYMS
Nolatrexed SCHEMBL18489 0.79 TYMS (0.66) TYMSDHFR
Nolatrexed SCHEMBL1649851 0.78 TYMS (0.65) TYMSDHFR
SCHEMBL16807869 0.75 TYMS (0.61) TYMSDHFR
SCHEMBL7827130 0.73 TYMS (1.00) TYMSDHFR
SCHEMBL7831197 0.72 TYMS (1.00) TYMSDHFR
SCHEMBL27555186 0.71 TYMS (0.58) TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105535991-A Amphiphilic basic group conjugate nanometer particles for treating tumors and preparation method thereof UNIV SHANGHAI JIAOTONG 2016-05-04 CN claimed
CN-112703004-B Methods and compositions for cancer treatment using recombinant dendritic cells 雷诺瓦罗生物制药公司 2025-02-14 CN disclosed
CN-112703004-A Methods and compositions for cancer treatment using recombinant dendritic cells 伊诺奇安生物制药公司 2021-04-23 CN disclosed
CN-105092752-B A kind of with liquid chromatography separation nolatrexed dihydrochloride and the method about material 北京康辰药业股份有限公司 2017-03-01 CN disclosed
CN-103298818-B Spiro-oxindole MDM2 antagonist 密歇根大学董事会 2016-06-29 CN disclosed
CN-105535991-A Amphiphilic basic group conjugate nanometer particles for treating tumors and preparation method thereof UNIV SHANGHAI JIAOTONG 2016-05-04 CN disclosed
CN-104619352-A Compositions containing hc-ha/ptx3 complexes and methods of use thereof TISSUETECH INC 2015-05-13 CN disclosed
CN-103282025-A Melt-extruded solid dispersions containing apoptosis-inducing agents ABBVIE INC 2013-09-04 CN disclosed