SCHEMBL27935552

SCHEMBL27935552

COc1ccnc(-c2cc(Nc3cccc4c3CCN(S(C)(=O)=O)C4)ccc2CN)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 7/20 0.36
MTOR P42345 3/20 0.35
PIK3CD O00329 2/20 0.35
PIK3CB P42338 2/20 0.35
PIK3CG P48736 2/20 0.35
PIK3C2B O00750 1/20 0.35
PIK3R1 P27986 1/20 0.35
PI4KB Q9UBF8 1/20 0.35
CHEK1 O14757 1/20 0.35
AURKA O14965 1/20 0.35
RPS6KA5 O75582 1/20 0.35
RPS6KA4 O75676 1/20 0.35
KIT P10721 1/20 0.35
RPS6KB1 P23443 1/20 0.35
CDK2 P24941 1/20 0.35
FLT3 P36888 1/20 0.35
RPS6KA3 P51812 1/20 0.35
RPS6KA2 Q15349 1/20 0.35
RPS6KA1 Q15418 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1921960 0.90 PIK3CA (0.36) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL27950026 0.89 NTRK1 (0.36) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL27935555 0.88 DGAT2 (0.37) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL27935551 0.86 KCNH2 (0.39) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL27935532 0.86 SCN9A (0.38) CHEK1AURKARPS6KA5RPS6KA4KIT
SCHEMBL27950065 0.86 PIK3CA (0.37) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL27935526 0.85 PIK3CA (0.35) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL27935539 0.83 PIK3CA (0.35) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL27935509 0.83 DGAT2 (0.38) SCN9AJAK2JAK3
SCHEMBL27935556 0.82 SCN9A (0.38) CHEK1AURKARPS6KA5RPS6KA4KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102203067-B Hedgehog pathway modulators IRM LLC 2014-01-15 CN claimed
CN-102203067-B Hedgehog pathway modulators IRM LLC 2014-01-15 CN disclosed