SCHEMBL27936741

SCHEMBL27936741

Cc1onc(-c2ccccc2F)c1C(=O)c1c(-c2ccccc2F)noc1C

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 7/20 0.62
EPAS1 Q99814 1/20 0.57
HSD17B10 Q99714 1/20 0.54
LMNA P02545 3/20 0.53
MAPT P10636 3/20 0.52
ALDH1A1 P00352 2/20 0.51
GAA P10253 2/20 0.50
PTGS1 P23219 1/20 0.50
TP53 P04637 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3826089 0.89 GPBAR1 (0.60) GPBAR1EPAS1HSD17B10LMNAMAPT
SCHEMBL2470614 0.89 GPBAR1 (0.60) GPBAR1EPAS1HSD17B10LMNAMAPT
SCHEMBL30395326 0.89 GPBAR1 (0.60) GPBAR1EPAS1HSD17B10LMNAMAPT
SCHEMBL3822684 0.88 HSD17B10 (0.70) GPBAR1EPAS1HSD17B10LMNAMAPT
SCHEMBL11408570 0.85 EPAS1 (0.61) GPBAR1EPAS1HSD17B10LMNAMAPT
SCHEMBL5773636 0.85 GPBAR1 (0.57) GPBAR1EPAS1HSD17B10LMNAMAPT
SCHEMBL2473847 0.84 GPBAR1 (0.56) GPBAR1EPAS1HSD17B10LMNAMAPT
SCHEMBL2924198 0.83 GPBAR1 (0.58) GPBAR1EPAS1LMNAMAPTALDH1A1
SCHEMBL27927955 0.83 HSD17B10 (0.55) GPBAR1EPAS1HSD17B10LMNAMAPT
SCHEMBL3976223 0.82 HTT (0.50) GPBAR1EPAS1HSD17B10LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103313982-A Phenyl-isoxazole derivatives and process for the preparation thereof IL YANG PHARM CO LTD 2013-09-18 CN claimed
CN-103313982-A Phenyl-isoxazole derivatives and process for the preparation thereof IL YANG PHARM CO LTD 2013-09-18 CN disclosed