SCHEMBL279452

SCHEMBL279452

CC(C)(C)OC(=O)N1C(=O)C(=Cc2ccc(F)c(Cl)c2)c2ccc(Cl)cc21

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.37
MAPT P10636 2/20 0.37
SNCA P37840 1/20 0.37
CYP3A4 P08684 2/20 0.35
CYP3A5 P20815 2/20 0.35
CNR1 P21554 2/20 0.35
PPARG P37231 1/20 0.35
CNR2 P34972 1/20 0.35
PAK1 Q13153 3/20 0.35
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
ERO1A Q96HE7 1/20 0.33
PIM1 P11309 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
GPR35 Q9HC97 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL274463 0.87 MDM4 (0.43) APPMAPTSNCACNR1PPARG
SCHEMBL274462 0.87 MDM4 (0.43) APPMAPTSNCACNR1PPARG
SCHEMBL277025 0.87 MDM4 (0.43) APPMAPTSNCACNR1PPARG
SCHEMBL279165 0.87 PPARG (0.45) APPMAPTSNCAPPARGMEN1
SCHEMBL275608 0.87 PPARG (0.45) APPMAPTSNCAPPARGMEN1
SCHEMBL275607 0.87 PPARG (0.45) APPMAPTSNCAPPARGMEN1
SCHEMBL275659 0.87 APP (0.35) APPMAPTSNCACYP3A4CYP3A5
SCHEMBL275658 0.87 APP (0.35) APPMAPTSNCACYP3A4CYP3A5
SCHEMBL275084 0.86 CYP3A4 (0.37) APPMAPTSNCACYP3A4CYP3A5
SCHEMBL275083 0.86 CYP3A4 (0.37) APPMAPTSNCACYP3A4CYP3A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8134001-B2 Spiroindolinone derivatives HOFFMANN-LA ROCHE INC. (US) 2012-03-13 US disclosed
WO-2009077357-A1 SPIROINDOLINONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-06-25 WO disclosed
US-20090156610-A1 Spiroindolinone Derivatives DING QINGJIE 2009-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156610-A1 Spiroindolinone Derivatives SDHA, AR, XPOT APP 4745/4885MAPT 4062/4885SNCA 480/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.