SCHEMBL27947682

SCHEMBL27947682

[CH2]CCc1ccc(NC(=O)OC(C)(C)C)nc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 2/20 0.48
HDAC1 Q13547 1/20 0.48
GRIN2B Q13224 1/20 0.44
CYP17A1 P05093 1/20 0.43
GSK3B P49841 1/20 0.41
DYRK1A Q13627 1/20 0.41
SCN9A Q15858 1/20 0.40
MAPKAPK2 P49137 2/20 0.39
BCL2 P10415 1/20 0.39
TSHR P16473 1/20 0.38
ATR Q13535 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
DEGS1 O15121 1/20 0.37
DRD2 P14416 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16296315 0.88 NAMPT (0.48) NAMPTHDAC1GRIN2BCYP17A1GSK3B
SCHEMBL8362974 0.88 HDAC1 (0.53) NAMPTHDAC1GRIN2BCYP17A1GSK3B
SCHEMBL13188545 0.86 NAMPT (0.47) NAMPTHDAC1GRIN2BCYP17A1GSK3B
SCHEMBL19669455 0.86 NAMPT (0.47) NAMPTHDAC1GRIN2BCYP17A1GSK3B
SCHEMBL30684527 0.86 P4HTM (0.48) NAMPTHDAC1GRIN2BCYP17A1GSK3B
SCHEMBL30684531 0.86 P4HTM (0.48) NAMPTHDAC1GRIN2BCYP17A1GSK3B
SCHEMBL540536 0.86 NAMPT (0.50) NAMPTHDAC1GRIN2BCYP17A1GSK3B
SCHEMBL15354526 0.86 NAMPT (0.50) NAMPTHDAC1GRIN2BCYP17A1GSK3B
SCHEMBL540467 0.84 NAMPT (0.49) NAMPTHDAC1GRIN2BCYP17A1GSK3B
SCHEMBL21394710 0.84 NAMPT (0.49) NAMPTHDAC1GRIN2BCYP17A1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102656163-B Suppress the heterogeneous ring compound of PASK BIOENERGENIX (US) 2016-01-13 CN claimed
CN-103459382-A Heterocyclic compounds for the inhibition of pask BIOENERGENIX LLC 2013-12-18 CN claimed
CN-102656163-B Suppress the heterogeneous ring compound of PASK BIOENERGENIX (US) 2016-01-13 CN disclosed
CN-103459382-A Heterocyclic compounds for the inhibition of pask BIOENERGENIX LLC 2013-12-18 CN disclosed