SCHEMBL27950403

SCHEMBL27950403

CC(C)(C)OC(=O)C(C)(N)C1CCCCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.41
DGAT1 O75907 1/20 0.41
EPHX1 P07099 5/20 0.41
HPGD P15428 1/20 0.36
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
SSTR4 P31391 1/20 0.33
BTK Q06187 1/20 0.33
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
SIGMAR1 Q99720 1/20 0.32
EPHX2 P34913 1/20 0.32
CTSS P25774 1/20 0.31
CTSK P43235 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6597535 0.98 DGAT1 (0.42) GAADGAT1EPHX1HPGDHDAC4
SCHEMBL27566889 0.90 DGAT1 (0.40) GAADGAT1EPHX1HPGDBTK
Hydrochloric Acid SCHEMBL6600019 0.88 DGAT1 (0.39) GAADGAT1EPHX1HPGDBTK
SCHEMBL26698295 0.86 EPHX1 (0.40) GAADGAT1EPHX1HPGDHDAC4
SCHEMBL7352585 0.84 EPHX1 (0.43) GAAEPHX1SSTR4PDK1PDK2
SCHEMBL7352590 0.84 EPHX1 (0.43) GAAEPHX1SSTR4PDK1PDK2
SCHEMBL28770712 0.84 EPHX1 (0.43) GAAEPHX1SSTR4PDK1PDK2
SCHEMBL26698284 0.84 EPHX1 (0.38) GAADGAT1EPHX1HPGDBTK
Hydrochloric Acid SCHEMBL5194471 0.82 EPHX1 (0.42) GAAEPHX1SSTR4PDK1PDK2
Hydrochloric Acid SCHEMBL27712371 0.82 EPHX1 (0.42) GAAEPHX1SSTR4PDK1PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102746175-B Substituted pyrimidodiazepines useful as PLK1 inhibitors TAKAEDA CHEMICAL IND LTD 2014-01-15 CN disclosed