SCHEMBL27951997

SCHEMBL27951997

CC(=O)c1cccnc1S

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.45
ALDH1A1 P00352 4/20 0.45
TDP1 Q9NUW8 1/20 0.45
MAPT P10636 2/20 0.44
CYP3A4 P08684 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
BLM P54132 1/20 0.44
AGER Q15109 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
NAPRT Q6XQN6 2/20 0.42
LMNA P02545 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
P2RX7 Q99572 1/20 0.42
MYC P01106 1/20 0.40
KDM4C Q9H3R0 1/20 0.39
PARP1 P09874 1/20 0.39
PRKCI P41743 2/20 0.39
KMT2A Q03164 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
2-Mercaptonicotinic Acid SCHEMBL3070055 0.82 KDM4E (0.59) KDM4EALDH1A1TDP1MAPTCYP3A4
2-Mercaptonicotinic Acid SCHEMBL261186 0.81 KDM4E (0.63) KDM4EALDH1A1TDP1MAPTCYP3A4
2-Mercaptonicotinic Acid SCHEMBL29382089 0.81 KDM4E (0.63) KDM4EALDH1A1TDP1MAPTCYP3A4
SCHEMBL4620997 0.81 KDM4E (0.47) KDM4EALDH1A1TDP1MAPTCYP3A4
SCHEMBL13623669 0.80 PDK2 (0.44) KDM4EALDH1A1TDP1MAPTCYP3A4
2-Mercaptonicotinic Acid SCHEMBL30605292 0.79 KDM4E (0.61) KDM4EALDH1A1TDP1MAPTCYP3A4
SCHEMBL1326787 0.79 PARP1 (0.56) KDM4EALDH1A1TDP1MAPTCYP3A4
SCHEMBL21995771 0.79 SMN1; SMN2 (0.47) KDM4EALDH1A1TDP1MAPTCYP3A4
2-Mercaptonicotinic Acid SCHEMBL29181672 0.79 KDM4E (0.61) KDM4EALDH1A1TDP1MAPTCYP3A4
2-Mercaptonicotinic Acid SCHEMBL29105774 0.79 KDM4E (0.61) KDM4EALDH1A1TDP1MAPTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103626693-A A class of pleuromytilin derivatives, drug composition, synthesis methods and uses thereof SHANGHAI INST MATERIA MEDICA 2014-03-12 CN disclosed