SCHEMBL27951998

SCHEMBL27951998

O=C(c1cccnc1)c1ccccc1Br

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 1/20 0.53
KCNH2 Q12809 1/20 0.53
HPGD P15428 1/20 0.52
TSHR P16473 1/20 0.52
ALDH1A1 P00352 3/20 0.52
APP P05067 1/20 0.52
GAA P10253 1/20 0.52
HCAR3 P49019 1/20 0.52
HCAR2 Q8TDS4 1/20 0.52
HDAC1 Q13547 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
F7 P08709 1/20 0.50
F3 P13726 1/20 0.50
SARM1 Q6SZW1 1/20 0.50
SIRT2 Q8IXJ6 1/20 0.50
SIRT6 Q8N6T7 1/20 0.50
SIRT1 Q96EB6 1/20 0.50
SIRT3 Q9NTG7 1/20 0.50
SIRT5 Q9NXA8 1/20 0.50
SIRT4 Q9Y6E7 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22426419 0.81 ALDH1A1 (0.56) HPGDALDH1A1APPGAAHCAR3
SCHEMBL7289960 0.81 AKR1C3 (0.66) ALDH1A1APPGAAHCAR3HCAR2
SCHEMBL6950942 0.79 GAA (0.65) HPGDALDH1A1APPGAAHCAR3
SCHEMBL6770549 0.79 HPGD (0.59) HPGDALDH1A1APPGAAHCAR3
SCHEMBL3251235 0.79 ALDH1A1 (0.52) HPGDALDH1A1APPGAAHCAR3
SCHEMBL11637980 0.79 ATM (0.59) ALDH1A1APPGAAHCAR3HCAR2
SCHEMBL29913321 0.79 AKR1C3 (0.61) ALDH1A1GAAKMT2APOLB
SCHEMBL723657 0.79 AKR1C3 (0.61) ALDH1A1GAAKMT2APOLB
SCHEMBL1242243 0.79 ALDH1A1 (0.71) ALDH1A1APPGAAHCAR3HCAR2
SCHEMBL29915528 0.79 ALDH1A1 (0.71) ALDH1A1APPGAAHCAR3HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103626693-A A class of pleuromytilin derivatives, drug composition, synthesis methods and uses thereof SHANGHAI INST MATERIA MEDICA 2014-03-12 CN disclosed